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Product Overview

Product Code

TRC-A790030

CAS Number

68844-77-9

Product Format

Neat

Molecular Formula

C28 H31 F N4 O

Molecular Weight

458.57

API Family

Astemizole

Product Categories

TRC, Antihistamines, API Reference Standards & Research Materials, Agonist & antagonist analogues, Additional Cancer Bioactive Molecules, Additional Neuro Products, Neurotransmission, Epilepsy, Multiple Sclerosis, Stroke, Pain and Inflammation, Histamine receptors, Pharmaceutical, Veterinary Compound & Metabolite Reference Materials , Pharmaceutical and Veterinary Residue Reference Materials , Pharmaceutical Toxicology Reference Materials , Pharmaceutical and veterinary compounds and metabolites Reference Materials

Product Type

API

Purity

>95% (HPLC)

Documentation

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Product Information

Chemical Data

Analyte Name

Astemizole

CAS Number

68844-77-9

Molecular Formula

C28 H31 F N4 O

Molecular Weight

458.57

Accurate Mass

458.2482

SMILES

COc1ccc(CCN2CCC(CC2)Nc3nc4ccccc4n3Cc5ccc(F)cc5)cc1

InChI

InChI=1S/C28H31FN4O/c1-34-25-12-8-21(9-13-25)14-17-32-18-15-24(16-19-32)30-28-31-26-4-2-3-5-27(26)33(28)20-22-6-10-23(29)11-7-22/h2-13,24H,14-20H2,1H3,(H,30,31)

IUPAC

1-[(4-fluorophenyl)methyl]-N-[1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl]benzimidazol-2-amine

Product Data

Storage Temperature

+4°C

Shipping Temperature

Room Temperature

Country of Origin

CANADA

Product Type

API

Product Format

Neat

API Family

Astemizole

Purity

>95% (HPLC)

Product Description

Nonsedating-type histamine H1-receptor antagonist. Potential for combination therapy with antivancer drugs such as doxorubicin in resistant leukemia. Antihistaminic.

References: Wauquier, A., et al.: Eur. J. Pharmacol., 72, 245 (1981), Laduron, P.M., et al.: Mol. Pharmacol., 21, 294 (1982), Richards, D.M., et al.: Drugs, 28, 38 (1984), Al-Obaid, A.M., et al.: Anal. Profiles Drug Subs., 20, 173 (1991), Ishikawa, M., et al.: Biol. Pharm. Bull., 23, 112 (2000),

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